Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
DCN1-like protein 1 (Homo sapiens) | BDBM50245154 (CHEMBL4067795 | US11116757, No. A10) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
St. Jude Children's Research Hospital Curated by ChEMBL | Assay Description Binding affinity for Adenosine A1 receptor using N-[3H] cyclohexyladenosine in rat forebrain membranes | J Med Chem 61: 2694-2706 (2018) Article DOI: 10.1021/acs.jmedchem.7b01282 BindingDB Entry DOI: 10.7270/Q22V2JHZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 (Homo sapiens) | BDBM50245154 (CHEMBL4067795 | US11116757, No. A10) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | US Patent | n/a | n/a | 78.9 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description The TR-FRET assay is illustrated in FIG. 3A and FIG. 3B. The TR-FRET assay cocktail was prepared by mixing 50 nM Biotin-DCN1P, 20 nM AlexaFluor488 UB... | Citation and Details BindingDB Entry DOI: 10.7270/Q2736V2B | |||||||||||
More data for this Ligand-Target Pair |