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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50245700   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Epidermal growth factor receptor


(Homo sapiens (Human))		BDBM50245700
PNG
(CHEMBL4077349)
Show SMILES Brc1ccc(cc1)C(=O)Nn1c(nc2ccccc2c1=O)-c1ccccc1
Show InChI InChI=1S/C21H14BrN3O2/c22-16-12-10-15(11-13-16)20(26)24-25-19(14-6-2-1-3-7-14)23-18-9-5-4-8-17(18)21(25)27/h1-13H,(H,24,26)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
GoogleScholar
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CHEMBL
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 420n/an/an/an/an/an/a



R. C. Patel Institute of Pharmaceutical Education and Research

Curated by ChEMBL


Assay Description
Inhibition of human EGFR preincubated for 5 mins with substrate followed by ATP addition measured after 30 mins by HTRF method

Bioorg Med Chem 25: 2713-2723 (2017)


Article DOI: 10.1016/j.bmc.2017.03.039
BindingDB Entry DOI: 10.7270/Q2NP26TD
More data for this
Ligand-Target Pair