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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50247615   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histone acetyltransferase KAT2B


(Homo sapiens (Human))		BDBM50247615
PNG
(2-(3,4,5-trifluorophenyl)isothiazol-3(2H)-one | CH...)
Show SMILES Fc1cc(cc(F)c1F)-n1sccc1=O
Show InChI InChI=1S/C9H4F3NOS/c10-6-3-5(4-7(11)9(6)12)13-8(14)1-2-15-13/h1-4H
PDB
MMDB

NCI pathway
Reactome pathway
KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 3.10E+3n/an/an/an/an/an/a



Institute of Cancer Research

Curated by ChEMBL


Assay Description
Inhibition of GST-fused recombinant HAT PCAF expressed in Escherichia coli by filter assay

Bioorg Med Chem 17: 467-74 (2009)


Article DOI: 10.1016/j.bmc.2008.11.079
BindingDB Entry DOI: 10.7270/Q2H70GRB
More data for this
Ligand-Target Pair