Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-activating factor receptor (Cavia porcellus) | BDBM50366241 (CHEMBL297624 | L-652731) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
Sankyo Co. Ltd Curated by ChEMBL | Assay Description Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAF | J Med Chem 39: 5281-4 (1997) Article DOI: 10.1021/jm950640q BindingDB Entry DOI: 10.7270/Q2FF3T06 | |||||||||||
More data for this Ligand-Target Pair |