Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-activating factor acetylhydrolase (Homo sapiens (Human)) | BDBM50162136 (CHEMBL3792924) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | 185 | n/a | n/a | n/a | n/a | n/a |
ShanghaiTech University Curated by ChEMBL | Assay Description Binding affinity to human Lp-PLA2 by ITC assay | J Med Chem 59: 5115-20 (2016) Article DOI: 10.1021/acs.jmedchem.6b00282 BindingDB Entry DOI: 10.7270/Q23F4RMQ | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |