Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanin-concentrating hormone receptor 1 (Homo sapiens (Human)) | BDBM50150715 (4''-Fluoro-biphenyl-4-carboxylic acid (6-dimethyla...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 5.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Neurocrine Biosciences Inc. Curated by ChEMBL | Assay Description Displacement of [125I]MCH from human Melanin-concentrating hormone 1 (MCH1) receptor modified for optimal expression in HEK293 cells | Bioorg Med Chem Lett 15: 999-1004 (2005) Article DOI: 10.1016/j.bmcl.2004.12.036 BindingDB Entry DOI: 10.7270/Q21R6R9X | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanin-concentrating hormone receptor 1 (RAT) | BDBM50150715 (4''-Fluoro-biphenyl-4-carboxylic acid (6-dimethyla...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 8.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Takeda Chemical Industries, Ltd. Curated by PDSP Ki Database | Eur J Pharmacol 438: 129-35 (2002) Article DOI: 10.1016/s0014-2999(02)01314-6 BindingDB Entry DOI: 10.7270/Q2GX495R | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melanin-concentrating hormone receptor 1 (Homo sapiens (Human)) | BDBM50150715 (4''-Fluoro-biphenyl-4-carboxylic acid (6-dimethyla...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 38 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Cerep Curated by ChEMBL | Assay Description Displacement of [125I][Phe13, Tyr19]MCH from human recombinant MCHR1 expressed in CHO cells | Bioorg Med Chem Lett 17: 3754-9 (2007) Article DOI: 10.1016/j.bmcl.2007.04.012 BindingDB Entry DOI: 10.7270/Q26D5SP0 | |||||||||||
More data for this Ligand-Target Pair |