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Compile Data Set for Download or QSAR

Found 1 hit of ki for monomerid = 50243121   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Histamine H3 receptor


(Rattus norvegicus (rat))		BDBM50243121
PNG
(2-hydroxy-1-((3aR,6aR)-6-(4-(2-(pyrrolidin-1-yl)et...)
Show SMILES OCC(=O)N1C[C@@H]2CC=C([C@@H]2C1)c1ccc(CCN2CCCC2)cc1 |r,c:8|
Show InChI InChI=1S/C21H28N2O2/c24-15-21(25)23-13-18-7-8-19(20(18)14-23)17-5-3-16(4-6-17)9-12-22-10-1-2-11-22/h3-6,8,18,20,24H,1-2,7,9-15H2/t18-,20+/m0/s1
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Article
PubMed
 6n/an/an/an/an/an/an/an/a



Arena Pharmaceuticals

Curated by ChEMBL


Assay Description
Displacement of N-[3H]methylhistamine from histamine H3 receptor in rat cortex membrane

Bioorg Med Chem Lett 18: 4133-6 (2008)


Article DOI: 10.1016/j.bmcl.2008.05.086
BindingDB Entry DOI: 10.7270/Q2C82942
More data for this
Ligand-Target Pair