Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
1-alkyl-2-acetylglycerophosphocholine esterase (Sus scrofa) | BDBM50085496 (CHEMBL89162 | N*1*,N*1*-Diethyl-hexadecane-1,2-dia...) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Univ. de Valencia Curated by ChEMBL | Assay Description Inhibition of secretory PLA2 activity in porcine pancreas using [3H]-oleate labelled membranes at a concentration of 10 uM | Bioorg Med Chem Lett 10: 285-8 (2000) BindingDB Entry DOI: 10.7270/Q2ZC8239 | |||||||||||
More data for this Ligand-Target Pair |