Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
3-phosphoinositide-dependent protein kinase 1 (Homo sapiens (Human)) | BDBM92493 (Alkaloid 2) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories | Assay Description 1536-Well TR-Fret uHTS assay PDK1-tide1 peptide substrate. | J Biol Chem 285: 18838-46 (2010) Article DOI: 10.1074/jbc.M109.089946 BindingDB Entry DOI: 10.7270/Q2PV6J0B | |||||||||||
More data for this Ligand-Target Pair |