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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM50283930'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
5-hydroxytryptamine receptor 2A


(Rattus norvegicus (rat))		BDBM50283930
PNG
(2-[4-(1,1-Diphenyl-silolan-3-yl)-piperazin-1-yl]-p...)
Show SMILES C1C[Si](CC1N1CCN(CC1)c1ncccn1)(c1ccccc1)c1ccccc1
Show InChI InChI=1S/C24H28N4Si/c1-3-8-22(9-4-1)29(23-10-5-2-6-11-23)19-12-21(20-29)27-15-17-28(18-16-27)24-25-13-7-14-26-24/h1-11,13-14,21H,12,15-20H2
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PC cid
PC sid
UniChem
Article
n/an/a 80n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
In vitro binding affinity towards serotonin 5-HT2A receptor in rat cortical membranes using [3H]ketanserin as radioligand

Bioorg Med Chem Lett 4: 415-420 (1994)


Article DOI: 10.1016/0960-894X(94)80007-3
BindingDB Entry DOI: 10.7270/Q2HX1D6M
More data for this
Ligand-Target Pair