Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
5-hydroxytryptamine receptor 2B (Homo sapiens (Human)) | BDBM50531776 (CHEMBL4533952) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a |
CSIR-Central Drug Research Institute (CSIR-CDRI) Curated by ChEMBL | Assay Description Positive allosteric modulation of 5HT2B receptor (unknown origin) expressed in HEK293 cells co-expressing NFAT-RE assessed as increase in serotonin-i... | Eur J Med Chem 164: 499-516 (2019) Article DOI: 10.1016/j.ejmech.2018.12.070 BindingDB Entry DOI: 10.7270/Q2XS5ZW2 | |||||||||||
More data for this Ligand-Target Pair |