Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
AP-4 complex subunit sigma-1 (Homo sapiens (Human)) | BDBM484149 ((R)-4-ethyl-9-(4- fluorobenzyl)-2-methyl-1-oxa- 4,...) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | <100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ESTEVE PHARMACEUTICALS. S.A. US Patent | Assay Description To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N... | US Patent US10927128 (2021) BindingDB Entry DOI: 10.7270/Q28918ZF | |||||||||||
More data for this Ligand-Target Pair |