Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
ATPase family AAA domain-containing protein 2 (Homo sapiens (Human)) | BDBM50520627 (CHEMBL4536031) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 166 | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Curated by ChEMBL | Assay Description Induction of ATAD2 bromodomain (unknown origin) dimerization | J Med Chem 61: 9004-9029 (2018) Article DOI: 10.1021/acs.jmedchem.8b00378 BindingDB Entry DOI: 10.7270/Q2N301BF | |||||||||||
More data for this Ligand-Target Pair |