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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Activin receptor type-1 [147-509]' and Ligand = 'BDBM575184'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Activin receptor type-1 [147-509]


(Homo sapiens (Human))
BDBM575184
PNG
(US11459329, Example 58)
Show SMILES CCn1cnc(c1)-c1ccc2c(ccnc2n1)-c1cnc2cc(c(C)nn12)-c1ccc(CN2CCO[C@@H](C)C2)cc1 |r|
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a<1n/an/an/an/an/an/a


TBA

Assay Description
ALK2 (aa 147-end) was obtained from BPS biosciences. The enzymatic assays were conducted in white 384-well polystyrene plates in a final volume of 8 ...


Citation and Details

BindingDB Entry DOI: 10.7270/Q2RJ4NQR
More data for this
Ligand-Target Pair