Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM50117223 (5-Butyl-8-(4-methoxy-phenyl)-3H-[1,2,4]triazolo[5,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 398 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Nutrition Research Institute Curated by ChEMBL | Assay Description Inhibition of [3H]-DPCPX binding to human Adenosine A1 receptor expressed in CHO cells; Range 256-620 | J Med Chem 45: 3703-8 (2002) BindingDB Entry DOI: 10.7270/Q2154GCW | |||||||||||
More data for this Ligand-Target Pair |