Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM50125912 (2-Furan-2-yl-8-methyl-9-methylsulfanyl-8H-pyrazolo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 8.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]- DPCPX binding at human Adenosine A1 receptor expressed in CHO cells | J Med Chem 46: 1229-41 (2003) Article DOI: 10.1021/jm021023m BindingDB Entry DOI: 10.7270/Q28916KP | |||||||||||
More data for this Ligand-Target Pair |