Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50212799 (9-benzyl-1,3-dimethyl-6,7,8,9-tetrahydropyrimido[1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.58E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Jagiellonian University Curated by ChEMBL | Assay Description Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane | Bioorg Med Chem 15: 5003-17 (2007) Article DOI: 10.1016/j.bmc.2007.04.018 BindingDB Entry DOI: 10.7270/Q2833RR7 | |||||||||||
More data for this Ligand-Target Pair |