Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Adenosine receptor A1 (Rattus norvegicus (rat)) | BDBM50366575 (CHEMBL609645) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Griffith University Curated by ChEMBL | Assay Description Binding affinity against adenosine A1 receptor in rat brain using [3H]R-PIA | Bioorg Med Chem Lett 8: 691-4 (1999) BindingDB Entry DOI: 10.7270/Q21Z44Z9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine receptor A1 (Homo sapiens (Human)) | BDBM50366575 (CHEMBL609645) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 1.00E+5 | n/a | n/a | n/a | n/a |
Griffith University Curated by ChEMBL | Assay Description Binding against Human Adenosine A1 receptor | Bioorg Med Chem Lett 8: 691-4 (1999) BindingDB Entry DOI: 10.7270/Q21Z44Z9 | |||||||||||
More data for this Ligand-Target Pair |