Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Adenosine receptor A2a (Rattus norvegicus (rat)) | BDBM110149 ((E)-8-(4-Bromostyryl)-1,3-diethyl-7-methylxanthine...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 28.9 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
North-West University, Private Bag X6001, Potchefstroom 2520, South Africa | Bioorg Chem 49: 49-58 (2013) Article DOI: 10.1016/j.bioorg.2013.06.006 BindingDB Entry DOI: 10.7270/Q21V5CM2 | ||||||||||||
More data for this Ligand-Target Pair |