Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Adenosine receptor A2a (Homo sapiens (Human)) | BDBM50451381 (CHEMBL38779) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | n/a | 0 | n/a | n/a | n/a | n/a |
University of Virginia Curated by ChEMBL | Assay Description AE maximal score at Adenosine A2A receptor | Bioorg Med Chem Lett 12: 1563-6 (2002) BindingDB Entry DOI: 10.7270/Q2833RBV | |||||||||||
More data for this Ligand-Target Pair |