Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Alpha-enolase (Homo sapiens (Human)) | BDBM50543109 (CHEMBL4647387) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 5.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.2c01039 BindingDB Entry DOI: 10.7270/Q2348QCK | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-enolase (Homo sapiens (Human)) | BDBM50543109 (CHEMBL4647387) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Texas MD Anderson Cancer Center Curated by ChEMBL | Assay Description Inhibition of ENO1 in overexpressed human D423 cells incubated for 5 days by crystal violet staining based spectrophotometry | ACS Med Chem Lett 11: 1484-1489 (2020) Article DOI: 10.1021/acsmedchemlett.0c00203 BindingDB Entry DOI: 10.7270/Q2SB499G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-enolase (Homo sapiens (Human)) | BDBM50543109 (CHEMBL4647387) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Texas MD Anderson Cancer Center Curated by ChEMBL | Assay Description Inhibition of ENO1 in wild-type human LN319 cells incubated for 5 days by crystal violet staining based spectrophotometry | ACS Med Chem Lett 11: 1484-1489 (2020) Article DOI: 10.1021/acsmedchemlett.0c00203 BindingDB Entry DOI: 10.7270/Q2SB499G | |||||||||||
More data for this Ligand-Target Pair |