Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Androgen receptor [646-919] (Homo sapiens (Human)) | BDBM227647 (HDSKGQTKLLQLLTTKSDQM | SCR-2 peptide) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.80E+3 | n/a | n/a | n/a | 6.5 | n/a |
Karlsruhe Institute of Technology | Assay Description For the fluorescence polarization experiments, 5 nM fluorescently labeled Bag-1L (Bag-1L(1-20), fluorescein isothiocyanate (FITC)-MAQRGGARRPRGDRERLGS... | J Biol Chem 289: 8839-51 (2014) Article DOI: 10.1074/jbc.M113.534859 BindingDB Entry DOI: 10.7270/Q2QZ28TM | |||||||||||
More data for this Ligand-Target Pair |