Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Angiopoietin-1 receptor (Homo sapiens (Human)) | BDBM50311970 (1-(3-(5-(4-aminothieno[2,3-d]pyrimidin-6-yl)-1-met...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Curated by ChEMBL | Assay Description Inhibition of Tie-2 phosphorylation by cell based assay | Bioorg Med Chem Lett 19: 6670-4 (2009) Article DOI: 10.1016/j.bmcl.2009.10.001 BindingDB Entry DOI: 10.7270/Q2FN16BJ | |||||||||||
More data for this Ligand-Target Pair |