Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Aromatase (Homo sapiens (Human)) | BDBM50104887 (2,3-dihydro-7-hydroxy-2-phenyl-4H-1-benzopyran-4-o...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 4021 Biomol�cules et Th�rapies anti-tumorales Curated by ChEMBL | Assay Description Inhibition of human aromatase in placental microsomes | Bioorg Med Chem 16: 1474-80 (2008) Article DOI: 10.1016/j.bmc.2007.10.057 BindingDB Entry DOI: 10.7270/Q2DR2WCC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50104887 (2,3-dihydro-7-hydroxy-2-phenyl-4H-1-benzopyran-4-o...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
UPRES EA 1085 Curated by ChEMBL | Assay Description Inhibition of aromatase activity in human placental microsomes | Bioorg Med Chem Lett 12: 2859-61 (2002) BindingDB Entry DOI: 10.7270/Q2PK0FHS | |||||||||||
More data for this Ligand-Target Pair |