Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
B-cell CLL/lymphoma 9 protein (Homo sapiens) | BDBM50577912 (CHEMBL4852661) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 5.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of C-terminal 6-His-tagged beta-catenin (1 to 781 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-N-terminal biotinyla... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00742 BindingDB Entry DOI: 10.7270/Q2SN0DSK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B-cell CLL/lymphoma 9 protein (Homo sapiens) | BDBM50577912 (CHEMBL4852661) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of C-terminal 6-His-tagged beta-catenin (1 to 781 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-N-terminal biotinyla... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c00742 BindingDB Entry DOI: 10.7270/Q2SN0DSK | |||||||||||
More data for this Ligand-Target Pair |