Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Beta-3 adrenergic receptor (Rattus norvegicus) | BDBM50193804 ((S)-6-(4-(2-(3-(3-(2-cyclobutylethyl)-2-oxo-2,3-di...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 29 | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at rat beta-3 adrenergic receptor expressed in CHO cells assessed as cAMP levels | Bioorg Med Chem Lett 16: 5691-4 (2006) Article DOI: 10.1016/j.bmcl.2006.08.010 BindingDB Entry DOI: 10.7270/Q2251HVR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-3 adrenergic receptor (Homo sapiens (Human)) | BDBM50193804 ((S)-6-(4-(2-(3-(3-(2-cyclobutylethyl)-2-oxo-2,3-di...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 10 | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at human beta3 adrenergic receptor expressed in CHO cells assessed as cAMP levels | Bioorg Med Chem Lett 16: 5691-4 (2006) Article DOI: 10.1016/j.bmcl.2006.08.010 BindingDB Entry DOI: 10.7270/Q2251HVR | |||||||||||
More data for this Ligand-Target Pair |