Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bombesin receptor subtype-3 (Homo sapiens (Human)) | BDBM50314966 (3-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 560 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation counting | Bioorg Med Chem Lett 20: 2074-7 (2010) Article DOI: 10.1016/j.bmcl.2010.02.076 BindingDB Entry DOI: 10.7270/Q2XW4JX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50314966 (3-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 97 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay relative to D-Tyr6-betaAla1... | Bioorg Med Chem Lett 20: 2074-7 (2010) Article DOI: 10.1016/j.bmcl.2010.02.076 BindingDB Entry DOI: 10.7270/Q2XW4JX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Mus musculus) | BDBM50314966 (3-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 14 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2074-7 (2010) Article DOI: 10.1016/j.bmcl.2010.02.076 BindingDB Entry DOI: 10.7270/Q2XW4JX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Homo sapiens (Human)) | BDBM50314966 (3-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.26E+3 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at human BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay | Bioorg Med Chem Lett 20: 2074-7 (2010) Article DOI: 10.1016/j.bmcl.2010.02.076 BindingDB Entry DOI: 10.7270/Q2XW4JX6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bombesin receptor subtype-3 (Homo sapiens (Human)) | BDBM50314966 (3-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 95 | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Agonist activity at human BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay relative to D-Tyr6-betaAla1... | Bioorg Med Chem Lett 20: 2074-7 (2010) Article DOI: 10.1016/j.bmcl.2010.02.076 BindingDB Entry DOI: 10.7270/Q2XW4JX6 | |||||||||||
More data for this Ligand-Target Pair |