Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bromodomain-containing protein 4 [44-166,I246A] (Homo sapiens (Human)) | BDBM227644 (Histone H4 (1-25) | MSGRGKGGKGLGKGGAKRHRKVLRD) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 1.71E+4 | n/a | n/a | n/a | 7.5 | 4 |
Bayer HealthCare | Assay Description The experiments were performed in 384-well black small volume microtiter plates(Greiner) in a buffer composed of 50mM Hepes, pH 7.5 (Applichem), 50 m... | J Biol Chem 289: 9304-19 (2014) Article DOI: 10.1074/jbc.M113.523019 BindingDB Entry DOI: 10.7270/Q2VQ31JB | |||||||||||
More data for this Ligand-Target Pair |