BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50256272'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Cannabinoid receptor 1 (Homo sapiens (Human))	BDBM50256272 (2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	48.9	n/a	n/a	n/a	n/a	n/a	n/a
National Central University Curated by ChEMBL					Assay Description Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cells				Bioorg Med Chem Lett 19: 1022-5 (2009) Article DOI: 10.1016/j.bmcl.2008.11.029 BindingDB Entry DOI: 10.7270/Q2Z89C8M
National Central University Curated by ChEMBL					More data for this Ligand-Target Pair
Cannabinoid receptor 1 (Homo sapiens (Human))	BDBM50256272 (2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...) Show SMILES Show InChI	PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	n/a	12.2	n/a	n/a	n/a	n/a
National Central University Curated by ChEMBL					Assay Description Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP binding				Bioorg Med Chem Lett 19: 1022-5 (2009) Article DOI: 10.1016/j.bmcl.2008.11.029 BindingDB Entry DOI: 10.7270/Q2Z89C8M
National Central University Curated by ChEMBL					More data for this Ligand-Target Pair