Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Casein kinase II subunit alpha (Homo sapiens (Human)) | BDBM15211 (CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 1.37E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute for Biochemistry Curated by ChEMBL | Assay Description Inhibitory constant against bovine CK2 | J Biol Chem 271: 26157-64 (1996) BindingDB Entry DOI: 10.7270/Q2BR8T3M | |||||||||||
More data for this Ligand-Target Pair |