Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor (Homo sapiens (Human)) | BDBM50000766 (CHEMBL12 | DIAZEPAM | US9271961, Diazepam) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Sharp& Dohme Research Laboratories Curated by ChEMBL | Assay Description Half-maximal inhibition of [125I]-CCK-8(+) binding to cholecystokinin receptor from guinea pig brain tissue | J Med Chem 31: 2235-46 (1989) BindingDB Entry DOI: 10.7270/Q2PG1S9K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor (RAT) | BDBM50000766 (CHEMBL12 | DIAZEPAM | US9271961, Diazepam) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptor | J Med Chem 30: 1229-39 (1987) BindingDB Entry DOI: 10.7270/Q2SF2WS2 | |||||||||||
More data for this Ligand-Target Pair |