Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cholecystokinin receptor type A (Cavia porcellus) | BDBM50046116 (3-(2-Amino-3-naphthalen-1-yl-propionylamino)-N-{1-...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
INSERM Curated by ChEMBL | Assay Description Displacement of [3H]-pCCK-8 from cholecystokinin-A receptor in guinea pig pancreatic membrane | J Med Chem 36: 166-72 (1993) BindingDB Entry DOI: 10.7270/Q26M37FJ | |||||||||||
More data for this Ligand-Target Pair |