Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cholecystokinin receptor type A (Mus musculus) | BDBM50287252 (3-{2-[2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3-dihy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibitory activity against Cholecystokinin type A receptor | Bioorg Med Chem Lett 6: 1421-1426 (1996) Article DOI: 10.1016/S0960-894X(96)00248-X BindingDB Entry DOI: 10.7270/Q2251J56 | |||||||||||
More data for this Ligand-Target Pair |