BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Cholesteryl ester transfer protein' and Ligand = 'BDBM50334826'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Cholesteryl ester transfer protein (Homo sapiens (Human))	BDBM50334826 (2-(4-(4-chlorophenyl)piperazin-1-yl)-N-(4-(5-cyano...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	53	n/a	n/a	n/a	n/a	n/a	n/a
Merck Research Laboratories Curated by ChEMBL					Assay Description Inhibition of human recombinant CETP-mediated cholesteryl ester transfer by fluorescence-based assay				Bioorg Med Chem Lett 21: 558-61 (2010) Article DOI: 10.1016/j.bmcl.2010.10.062 BindingDB Entry DOI: 10.7270/Q2XK8FT1
Merck Research Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair
Cholesteryl ester transfer protein (Homo sapiens (Human))	BDBM50334826 (2-(4-(4-chlorophenyl)piperazin-1-yl)-N-(4-(5-cyano...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	135	n/a	n/a	n/a	n/a	n/a	n/a
Merck Research Laboratories Curated by ChEMBL					Assay Description Inhibition of human recombinant CETP-mediated triglyceride transfer by fluorescence-based assay				Bioorg Med Chem Lett 21: 558-61 (2010) Article DOI: 10.1016/j.bmcl.2010.10.062 BindingDB Entry DOI: 10.7270/Q2XK8FT1
Merck Research Laboratories Curated by ChEMBL					More data for this Ligand-Target Pair