Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Choline kinase alpha (Homo sapiens (Human)) | BDBM50556491 (CHEMBL4784458) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.74E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human CKalpha1 assessed as reduction in 14C incorporation from [methyl-14C]choline to phosphatidylcholine using [methyl-14C]choline as ... | Citation and Details Article DOI: 10.1016/j.ejmech.2020.112797 BindingDB Entry DOI: 10.7270/Q25X2DKT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Choline kinase alpha (Homo sapiens (Human)) | BDBM50556491 (CHEMBL4784458) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 370 | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometry | Citation and Details Article DOI: 10.1016/j.ejmech.2020.112797 BindingDB Entry DOI: 10.7270/Q25X2DKT | |||||||||||
More data for this Ligand-Target Pair |