Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cholinesterase (Equus caballus (Horse)) | BDBM50402590 (CHEMBL2205576) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University College of Science Curated by ChEMBL | Assay Description Inhibition of equine serum BuChE using acetylthiocholine iodide as substrate by Ellman's method | Bioorg Med Chem 20: 7214-22 (2012) Article DOI: 10.1016/j.bmc.2012.08.052 BindingDB Entry DOI: 10.7270/Q2SQ91J0 | |||||||||||
More data for this Ligand-Target Pair |