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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Cyclic AMP-dependent transcription factor ATF-4' and Ligand = 'BDBM524127'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Cyclic AMP-dependent transcription factor ATF-4


(Human)
BDBM524127
PNG
(US11166942, Compound 16)
Show SMILES Fc1cc(OCCCN2CCN(CC2)NC(=O)COc2ccc(Cl)c(F)c2)ccc1Cl
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 125n/an/an/an/an/an/a


TBA

Assay Description
The ATF4 reporter was prepared by fusing the human full length 5′UTR of ATF4 (NCBI Accession No. BC022088.2) upstream of the firefly luciferase...


Citation and Details

BindingDB Entry DOI: 10.7270/Q2QJ7MG1
More data for this
Ligand-Target Pair