Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3 (Homo sapiens (Human)) | BDBM50088619 (2-(2-Fluoro-phenyl)-5,7-dihydroxy-8-(1-methyl-1,2,...) | PDB UniProtKB/SwissProt antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitotix Inc. Curated by ChEMBL | Assay Description Inhibitory activity against cyclin-dependent kinase 4-cyclin D1 | Bioorg Med Chem Lett 10: 1037-41 (2000) BindingDB Entry DOI: 10.7270/Q2959J22 | |||||||||||
More data for this Ligand-Target Pair |