Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cyclin-dependent kinase 5 activator 1 (Homo sapiens (Human)) | BDBM50499138 (CHEMBL3735368) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Fran£ois-Rabelais de Tours Curated by ChEMBL | Assay Description Inhibition of human recombinant CDK5/P25 expressed in Escherichia coli using histone H1 substrate after 30 mins by scintillation and luminescence cou... | Eur J Med Chem 105: 80-105 (2015) Article DOI: 10.1016/j.ejmech.2015.10.004 BindingDB Entry DOI: 10.7270/Q2736TX4 | |||||||||||
More data for this Ligand-Target Pair |