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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Cysteinyl leukotriene receptor 1/2' and Ligand = 'BDBM50057239'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Cysteinyl leukotriene receptor 1/2


(Homo sapiens (Human))		BDBM50057239
PNG
(2-Hydroxy-5-methyl-3-{(E)-3-[3-((E)-2-quinolin-2-y...)
Show SMILES Cc1cc(C(O)=O)c(O)c(c1)C(=O)\C=C\c1cccc(\C=C\c2ccc3ccccc3n2)c1
Show InChI InChI=1S/C28H21NO4/c1-18-15-23(27(31)24(16-18)28(32)33)26(30)14-10-20-6-4-5-19(17-20)9-12-22-13-11-21-7-2-3-8-25(21)29-22/h2-17,31H,1H3,(H,32,33)/b12-9+,14-10+
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Similars
Article
PubMed
n/an/an/a 105n/an/an/an/an/a



Vrije Universiteit

Curated by ChEMBL


Assay Description
Displacement of [3H]LTD4 from Cysteinyl leukotriene D4 receptor in guinea pig lung membranes

J Med Chem 40: 1075-89 (1997)


Article DOI: 10.1021/jm960628d
BindingDB Entry DOI: 10.7270/Q25141XJ
More data for this
Ligand-Target Pair