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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Cytosol aminopeptidase [33-68,L62W]' and Ligand = 'BDBM234296'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Cytosol aminopeptidase [33-68,L62W]


(Sus scrofa (Pig))
BDBM234296
PNG
(Nle-PH (4))
Show SMILES CCCCC(N)P(O)=O
Show InChI InChI=1S/C5H14NO2P/c1-2-3-4-5(6)9(7)8/h5,9H,2-4,6H2,1H3,(H,7,8)
UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
7.39E+4 -23.6n/an/an/an/an/a8.425



Academy of Sciences of the Czech Republic



Assay Description
LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was...


J Enzyme Inhib Med Chem 26: 155-61 (2011)


Article DOI: 10.3109/14756366.2010.482047
BindingDB Entry DOI: 10.7270/Q22N515B
More data for this
Ligand-Target Pair