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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'D(1A) dopamine receptor' and Ligand = 'BDBM50282001'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
D(1A) dopamine receptor


(RAT)		BDBM50282001
PNG
((4,5-Dihydro-3H-pyrazolo[4,5,1-ij]quinolin-4-yl)-d...)
Show SMILES CCCN(CCC)C1Cc2cnn3cccc(C1)c23
Show InChI InChI=1S/C16H23N3/c1-3-7-18(8-4-2)15-10-13-6-5-9-19-16(13)14(11-15)12-17-19/h5-6,9,12,15H,3-4,7-8,10-11H2,1-2H3
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars
Article
n/an/a>1.00E+5n/an/an/an/an/an/a



TBA

Curated by ChEMBL


Assay Description
Compound was evaluated for binding affinity to Dopamine receptor D1 labeled with [3H]-SCH- 23390 (0.3 nM) in rat striatal membranes

Bioorg Med Chem Lett 3: 1477-1483 (1993)


Article DOI: 10.1016/S0960-894X(00)80003-7
BindingDB Entry DOI: 10.7270/Q2MS3T7B
More data for this
Ligand-Target Pair