Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
D(3) dopamine receptor (Homo sapiens (Human)) | BDBM50339685 (4-(Thiophen-3-yl)-N-(4-(4-(2-(2-fluoroethoxy)pheny...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.170 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Washington University School of Medicine Curated by ChEMBL | Assay Description Displacement of [125I]-IABN from human D3 receptor transfected in human HEK 293 cells by gamma-counting | J Med Chem 54: 1555-64 (2011) Article DOI: 10.1021/jm101323b BindingDB Entry DOI: 10.7270/Q2WD40W0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(3) dopamine receptor (Homo sapiens (Human)) | BDBM50339685 (4-(Thiophen-3-yl)-N-(4-(4-(2-(2-fluoroethoxy)pheny...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 28 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Temple University School of Pharmacy Curated by ChEMBL | Assay Description Displacement of 2,3-dimethoxy-5-[125I]-iodo-N-[9-benzyl-9-azabicyclo[3.3.1]nonan-3beta-yl]benzamide from human dopamine D3 receptor expressed in HEK2... | Bioorg Med Chem Lett 29: 2690-2694 (2019) Article DOI: 10.1016/j.bmcl.2019.07.020 BindingDB Entry DOI: 10.7270/Q2JQ14CS | |||||||||||
More data for this Ligand-Target Pair |