Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Diacylglycerol O-acyltransferase 1 (Homo sapiens (Human)) | BDBM50499973 (CHEMBL3740607) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 57 | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi-aventis R&D Curated by ChEMBL | Assay Description Inhibition of recombinant human DGAT-1 using 1,2,di(cis-9-octadecenoyl)-sn-glycerol as substrate by Microbeta counter | Bioorg Med Chem Lett 26: 25-32 (2016) Article DOI: 10.1016/j.bmcl.2015.11.046 BindingDB Entry DOI: 10.7270/Q2Z89GDN | |||||||||||
More data for this Ligand-Target Pair |