Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Discoidin domain-containing receptor 2 (Homo sapiens (Human)) | BDBM163698 (5-((2-Methyl-5-((3-(4-methylpiperazin-1-yl)-5-(tri...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a | n/a |
Dana-Farber Cancer Institute | Assay Description The enzymatic activities DDR2 were tested in LanthaScreen binding assays. The protocol is available from Life Technologies. | ACS Chem Biol 10: 2687-96 (2015) Article DOI: 10.1021/acschembio.5b00655 BindingDB Entry DOI: 10.7270/Q2SX6BZ1 | |||||||||||
More data for this Ligand-Target Pair |