Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Dual specificity mitogen-activated protein kinase kinase 2 (Homo sapiens (Human)) | BDBM50387974 (CHEMBL2057830) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sejong University Curated by ChEMBL | Assay Description Inhibition of MEK2 using [gamma32P]ATP by radiometric kinase assay | Bioorg Med Chem Lett 22: 4946-50 (2012) Article DOI: 10.1016/j.bmcl.2012.06.041 BindingDB Entry DOI: 10.7270/Q25Q4X5B | |||||||||||
More data for this Ligand-Target Pair |