Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Dual specificity tyrosine-phosphorylation-regulated kinase 1A (RAT) | BDBM50295879 (4-(1-Methyl-1H-indol-3-yl)-5-(3-aminophenyl)pyrimi...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Clermont Universit£ Curated by ChEMBL | Assay Description Inhibition of rat recombinant DYRK1A expressed in Escherichia coli | Bioorg Med Chem 17: 4420-4 (2009) Article DOI: 10.1016/j.bmc.2009.05.017 BindingDB Entry DOI: 10.7270/Q2639PSH | |||||||||||
More data for this Ligand-Target Pair |