Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Dual specificity tyrosine-phosphorylation-regulated kinase 3 (Homo sapiens (Human)) | BDBM317462 (4-(4-(cyclopentyloxy)-5-(2- methylbenzo[d]oxazol-6...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 99 | n/a | n/a | n/a | n/a | n/a | n/a |
Celgene Corporation Curated by ChEMBL | Assay Description Inhibition of human full length recombinant GST-tagged DYRK3 expressed in baculovirus by Z'-LYTE assay | J Med Chem 60: 8989-9002 (2017) Article DOI: 10.1021/acs.jmedchem.7b01223 BindingDB Entry DOI: 10.7270/Q2GF0WX9 | |||||||||||
More data for this Ligand-Target Pair |