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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Ecdysone receptor (Choristoneura fumiferana) | BDBM50128305 (3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet  | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | n/a | n/a | 280 | n/a | n/a | n/a | n/a |
RHeoGene Curated by ChEMBL | Assay Description Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cells | Bioorg Med Chem Lett 13: 1883-6 (2003) BindingDB Entry DOI: 10.7270/Q2TM79HC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Ecdysone receptor (Bombyx mori) | BDBM50128305 (3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
RHeoGene Curated by ChEMBL | Assay Description Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK-293 cell-l... | Bioorg Med Chem Lett 13: 1883-6 (2003) BindingDB Entry DOI: 10.7270/Q2TM79HC | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Ecdysone receptor (Bombyx mori) | BDBM50128305 (3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 6 | n/a | n/a | n/a | n/a |
Ghent University Curated by ChEMBL | Assay Description Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assay | Pest Manag Sci 66: 1215-29 (2010) Article DOI: 10.1002/ps.1998 BindingDB Entry DOI: 10.7270/Q2FT8PXB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Ecdysone receptor (Bombyx mori) | BDBM50128305 (3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.40 | n/a | n/a | n/a | n/a |
Ghent University Curated by ChEMBL | Assay Description Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assay | Pest Manag Sci 66: 526-35 (2010) Article DOI: 10.1002/ps.1903 BindingDB Entry DOI: 10.7270/Q2KK9FPH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Ecdysone receptor (Spodoptera littoralis) | BDBM50128305 (3-methoxy-2-methylbenzoic acid 2-(3,5-dimethylbenz...) | PDB MMDB Reactome pathway KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 6 | n/a | n/a | n/a | n/a |
Ghent University Curated by ChEMBL | Assay Description Agonist activity at ecdysone receptor in Spodoptera littoralis Sl2 cells after 24 hr by luciferase reporter gene assay | Pest Manag Sci 66: 526-35 (2010) Article DOI: 10.1002/ps.1903 BindingDB Entry DOI: 10.7270/Q2KK9FPH | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
