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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Endoplasmic reticulum aminopeptidase 2' and Ligand = 'BDBM50170900'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Endoplasmic reticulum aminopeptidase 2


(Homo sapiens (Human))
BDBM50170900
PNG
(CHEMBL3806247)
Show SMILES CCCCCCNCC(N)P(O)(O)=O
Show InChI InChI=1/C8H21N2O3P/c1-2-3-4-5-6-10-7-8(9)14(11,12)13/h8,10H,2-7,9H2,1H3,(H2,11,12,13)
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PC cid
PC sid
UniChem
Article
PubMed
632n/an/an/an/an/an/an/an/a



Wroclaw University of Technology

Curated by ChEMBL


Assay Description
Inhibition of human ERAP2 preincubated for 30 to 60 mins followed by addition of Arg-AMC as substrate measured for 15 mins by spectrofluorimetric met...


Bioorg Med Chem Lett 26: 4122-6 (2016)


Article DOI: 10.1016/j.bmcl.2016.06.062
BindingDB Entry DOI: 10.7270/Q2TT4SW1
More data for this
Ligand-Target Pair